
Last Updated :2025/04/04
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Research activity information
Paper
- Cardo Bisphenol Fused with DIbenzo[g,p]chrysene for a High Refractive Index Monomer
Toko Yura; Rion Noda; Ikuma Okada; Zhenfeng Guo; Takashi Nakanishi; Yousuke Yamaoka; Tetsuo Iwasawa
European Journal of Organic Chemistry, Jan. 2025, [Reviewed] - Stable and Minimum Size Solubilization of Membrane Proteins with Cocktails of Phospholipid Analogues
Mai Takagi; Ayana Nagatani; Kenichi Kawano; Ayami Hata; Azusa Yokoyama; Koichi Hayashida; Haruka Hoshi; Mao Sakurai; Tsuyoshi Oyama; Yusuke Kuroda; Yousuke Yamaoka; Takahiro Fujiwara; Yohei Miyanoiri; Masaru Hoshino; Yoshiaki Yano; Kiyosei Takasu; Katsumi Matsuzaki
ACS Applied Materials & Interfaces, Nov. 2024 - Construction of Multiple Five-Membered Rings in Dibenzo[g,p]chrysene Core for the Synthesis of a Nona-cycle Buckybowl
Naruhiro Yoshida; Tomoya Imai; Toru Amaya; Yousuke Yamaoka; Tetsuo Iwasawa
European Journal of Organic Chemsitry, Sep. 2024, [Reviewed] - Chromic properties of dibenzo[j,l]fluoranthenes exhibiting different resonance contributions.
Kazuma Kurokawa; Naoki Ogawa; Yusuke Kuroda; Yousuke Yamaoka; Hiroshi Takikawa; Kazunori Tsubaki; Kiyosei Takasu
Organic & biomolecular chemistry, May 2024 - Intramolecular Cyclopropanation of Active Methylene Derivatives Based on FeCl2 or FeCl3‐Promoted Radical‐Polar Crossover Reactions
Eito Yoshioka; Yuuki Imoto; Yousuke Yamaoka; Tomoko Ikeda; Hiroki Takahashi; Ryousuke Tanaka; Naoki Hayashi; Hideto Miyabe
Chemistry – A European Journal, Apr. 2024 - NHC-Catalyzed Reaction of Aldehydes for C(sp2)–O Bond Formation
Yousuke Yamaoka; Hideto Miyabe
Catalysts, Mar. 2024 - Entry into Lithium Ynolates from α,α,α-Tribromomethyl Ketones: Synthesis of Cyclobutenes via the [2 + 2] Cycloaddition with α,β-Unsaturated Carbonyls
Yousuke Yamaoka; Hidetaka Imahori; Motoki Namioka; Ryo Nishina; Yukiko Kobori; Motoki Ueda; Mitsuru Shindo; Kiyosei Takasu
Organic Letters, Mar. 2024 - Total Synthesis of 1,4a-di-epi-ent-Pancratistatin, Exemplifying a Stereodivergent Approach to Pancratistatin Isomers
Chunzhao Sun; Tsubasa Inokuma; Daisuke Tsuji; Yousuke Yamaoka; Reiko Akagi; Ken-ichi Yamada
Chemical Communications, 2024 - 5-exo-Selective Asymmetric Bromolactonization of Stilbenecarboxylic Acids Catalyzed by Phenol-bearing Chiral Thiourea
Masayuki Sugano; Tsubasa Inokuma; Yousuke Yamaoka; Ken-ichi Yamada
Organic & Biomolecular Chemistry, 2024 - Regiocontrol Using Fluoro Substituent on 3,6-Disubstituted Arynes
Eito Yoshioka; Yousuke Yamaoka; Shunsuke Shimada; Hikaru Tanaka; Hideto Miyabe
Chemical and Pharmaceutical Bulletin, Oct. 2023 - Cross-Dimerization of Fluorenones for Synthesis of Dibenzo[g,p]chrysenes
Naruhiro Yoshida; Ryuhei Akasaka; Yousuke Yamaoka; Takafumi Yashima; Yuij Tokunaga; Tetsuo Iwasawa
Tetrahedron, Jul. 2023, [Reviewed] - Synthesis of an Octacyclic C60 Fragment
Naruhiro Yoshida; Ryuhei Akasaka; Tomoya Imai; Michael P. Schramm; Yousuke Yamaoka; Toru Amaya; Tetsuo Iwasawa
European Journal of Organic Chemistry, Jun. 2023, [Reviewed] - Rotaxane Synthesis by an End-Capping Strategy via Swelling Axle-Phenols.
Koki Fujimura; Yoshihiro Ueda; Yousuke Yamaoka; Kiyosei Takasu; Takeo Kawabata
Angewandte Chemie (International ed. in English), May 2023 - Efficient Synthesis of Medium‐sized Nitrogen Heterocycles by Brønsted Acid‐Catalyzed Cyclization of Ene‐ynamides
Yousuke Yamaoka; Nao Takeuchi; Ken‐ichi Yamada; Kiyosei Takasu
Asian Journal of Organic Chemistry, Apr. 2023 - Synthesis of γ-Aryl Medium-Sized Cyclic Enones by a Domino 4π-Electrocyclic Reaction/Heck–Matsuda Arylation Sequence at Ambient Temperature
Kiyosei Takasu; Tomohiro Ito; Nao Takeuchi; Yousuke Yamaoka; Hiroshi Takikawa
Synlett, Feb. 2023 - Remote electronic effect on the N-heterocyclic carbene-catalyzed asymmetric intramolecular Stetter reaction and structural revision of products
Tsubasa Inokuma; Kohei Iritani; Yuki Takahara; Chunzhao Sun; Yousuke Yamaoka; Satoru Kuwano; Ken-ichi Yamada
Chemical Communications, 2023 - Development of Antimicrobial Peptide-Antibiotic Conjugates to Improve the Outer Membrane Permeability of Antibiotics Against Gram-Negative Bacteria.
Ruka Yamauchi; Kenichi Kawano; Yousuke Yamaoka; Aoi Taniguchi; Yoshiaki Yano; Kiyosei Takasu; Katsumi Matsuzaki
ACS infectious diseases, Oct. 2022 - Lewis Acid-Catalyzed Diastereoselective Domino Reaction of Ene-Ynamide with Trimethylsilyl Cyanide to Construct Spiroindolines.
Yousuke Yamaoka; Daisuke Yamasaki; Daigo Kajiwara; Makiko Shinozaki; Ken-Ichi Yamada; Kiyosei Takasu
Organic letters, Jun. 2022 - Enhanced Molecular Recognition through Substrate–Additive Complex Formation in N-Heterocyclic-Carbene-Catalyzed Kinetic Resolution of α-Hydroxythioamides
Yinli Wang; Akiho Yamauchi; Keiji Hashimoto; Tatsuya Fujiwara; Tsubasa Inokuma; Yuta Mitani; Koichi Ute; Satoru Kuwano; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
ACS Catalysis, May 2022 - Relevant synthesis to manipulating non-planarity in dibenzo[g,p]chrysene: Substitution reactions at the bay
Shinsuke Kamiguchi; Ryuhei Akasaka; Naruhiro Yoshida; Tomoya Imai; Yousuke Yamaoka; Toru Amaya; Tetsuo Iwasawa
Tetrahedron Letters, Mar. 2022, [Reviewed] - Total Synthesis of Cryptopleurine and Its Analogues
Yousuke Yamaoka; Kiyosei Takasu; Takuro Yamakawa; Kaito Tateishi
Synthesis, Jan. 2022 - Oxidative β-Cleavage of Fused Cyclobutanols Leading to Hydrofuran-Fused Polycyclic Aromatic Compounds.
Hayate Kinouchi; Kazuma Sugimoto; Yousuke Yamaoka; Hiroshi Takikawa; Kiyosei Takasu
The Journal of organic chemistry, Sep. 2021 - The rationale for stereoinduction in conjugate addition to alkylidenemalonates bearing a menthol-derived chiral auxiliary
Ken-ichi Yamada; Shinichi Fujiwara; Tsubasa Inokuma; Masayuki Sugano; Yousuke Yamaoka; Kiyosei Takasu
Tetrahedron, Jul. 2021 - Mechanistic Support for Intramolecular Migrative Cyclization of Propargyl Sulfones Provided by Catalytic Asymmetric Induction with a Chiral Counter Cation Strategy
Kohta Yamasaki; Akiho Yamauchi; Tsubasa Inokuma; Yasunori Miyakawa; Yinli Wang; Raphaël Oriez; Yousuke Yamaoka; Kiyosei Takasu; Naonobu Tanaka; Yoshiki Kashiwada; Ken‐ichi Yamada
Asian Journal of Organic Chemistry, May 2021 - Synthesis of Lactone-Fused Cyclopropanes by Ring Contractive α-Ketol Rearrangement of Ketal-Fused Cyclobutanones
Kiyosei Takasu; Koichi Shigenaga; Kazuma Shimoda; Hiroshi Takikawa; Yousuke Yamaoka
HETEROCYCLES, 2021 - Total Synthesis of (-)-Sigillin A: A Polychlorinated and Polyoxygenated Natural Product.
Yousuke Yamaoka; Takamori Nakayama; Shota Kawai; Kiyosei Takasu
Organic letters, Oct. 2020 - Helical Nanographenes Embedded with Contiguous Azulene Units.
Naoki Ogawa; Yousuke Yamaoka; Hiroshi Takikawa; Ken-Ichi Yamada; Kiyosei Takasu
Journal of the American Chemical Society, Aug. 2020 - Helical Graphene Nanostructures Embedded with an Azulene Cluster
Yousuke Yamaoka; Naoki Ogawa; Hiroshi Takikawa; Ken-ichi Yamada; Kiyosei Takasu
Apr. 2020 - Helical Graphene Nanostructures Embedded with an Azulene Cluster
Yousuke Yamaoka; Naoki Ogawa; Hiroshi Takikawa; Ken-ichi Yamada; Kiyosei Takasu
Apr. 2020 - Synthesis of Dibenzoxazonines by Domino [2+2] Cycloaddition—4π Electrocyclic Ring Opening Reaction of Cyclic Imines with Ynamides
Kiyosei Takasu; Masaki Tsutsumi; Tomohiro Ito; Hiroshi Takikawa; Yousuke Yamaoka
HETEROCYCLES, 2020, [Reviewed] - Synthesis of Polycyclic Spirocarbocycles via Acid-Promoted Ring-Contraction/Dearomative Ring-Closure Cascade of Oxapropellanes.
Ogawa N; Yamaoka Y; Takikawa H; Takasu K
Organic letters, Sep. 2019, [Reviewed] - Total Syntheses of Allelopathic 4-Oxyprotoilludanes, Melleolides, and Echinocidins.
Shimoda K; Yamaoka Y; Yoo D; Yamada KI; Takikawa H; Takasu K
The Journal of organic chemistry, Sep. 2019, [Reviewed] - Synthesis of Functionalized Medium-Sized trans-Cycloalkenes by 4π Electrocyclic Ring Opening-Alkylation Cascade.
Takasu K; Ito T; Tsutsumi M; Yamada KI; Takikawa H; Yamaoka Y
Angewandte Chemie (International ed. in English), Jul. 2019, [Reviewed] - Rapid Assembly of Protoilludane Skeleton through Tandem Catalysis: Total Synthesis of Paesslerin A and Its Structural Revision
Y. Mogi; K. Inanaga; H. Tokuyama; M. Ihara; Y. Yamaoka; K. Yamada; K. Takasu
Organic Letters, 2019, [Reviewed] - Optical resolution via catalytic generation of chiral auxiliary
Hiroki Kiyama; Tsubasa Inokuma; Yusuke Kuroda; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
Tetrahedron Letters, Jan. 2019, [Reviewed] - Silyl enol etherification by a Tf
2 NH/amine co-catalytic system for minimizing hazardous waste generation
Kei Kurahashi; Yousuke Yamaoka; Yoshiji Takemoto; Kiyosei Takasu
Reaction Chemistry and Engineering, Oct. 2018, [Reviewed] - Synthesis and Properties of Tribenzocarbazoles via an Acid-promoted Retro (2+2)-Cycloaddition of Azapropellanes
Naoki Ogawa; Yousuke Yamaoka; Hiroshi Takikawa; Kazunori Tsubaki; Kiyosei Takasu
Journal of Organic Chemistry, 2018, [Reviewed] - Total Synthesis of Phenanthroquinolizidine Alkaloid Cryptopleurine and Phenanthroindolizidine Alkaloid Tylophorine
Yohsuke Yamaoka
Heteroccycles, 2018, [Reviewed] - Synthesis and biological evaluation of steroidal derivatives bearing a small ring as vitamin D receptor agonists
Norihito Arichi; Shinichi Fujiwara; Michiyasu Ishizawa; Makoto Makishima; Duy H. Hua; Ken-ichi Yamada; Yousuke Yamaoka; Kiyosei Takasu
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, Aug. 2017, [Reviewed] - Synthesis of multi-substituted cyclobutenes: Cyclic strategy for [2+2] cycloaddition of ketene silyl acetals with propiolates
Yousuke Yamaoka; Motoki Ueda; Tohru Yamashita; Kazuma Shimoda; Ken-ichi Yamada; Kiyosei Takasu
TETRAHEDRON LETTERS, Jul. 2017, [Reviewed] - Synthesis of pi-Extended Fluoranthenes via a KHMDS-Promoted Anionic-Radical Reaction Cascade
Naoki Ogawa; Yousuke Yamaoka; Ken-ichi Yamada; Kiyosei Takasu
ORGANIC LETTERS, Jun. 2017, [Reviewed] - Site-selective benzoin-type cyclization of unsymmetrical dialdoses catalyzed by N-heterocyclic carbenes for divergent cyclitol synthesis
Bubwoong Kang; Yinli Wang; Satoru Kuwano; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
CHEMICAL COMMUNICATIONS, Apr. 2017, [Reviewed] - PHOSPHINE-PROMOTED MIGRATIVE CYCLIZATION OF SULFONYLALKYNOL AND SULFONYLALKYNAMIDE FOR THE SYNTHESIS OF OXA- AND AZACYCLES
Yinli Wang; Raphael Oriez; Shougun Ou; Yasunori Miyakawa; Yousuke Yamaoka; Kiyosei Takasu; Ken-Ichi Yamada
HETEROCYCLES, Jan. 2017, [Reviewed] - Use of a Catalytic Chiral Leaving Group for Asymmetric Substitutions at sp(3)-Hybridized Carbon Atoms: Kinetic Resolution of beta-Amino Alcohols by p-Methoxybenzylation
Yusuke Kuroda; Shingo Harada; Akinori Oonishi; Hiroki Kiyama; Yousuke Yamaoka; Ken-ichi Yamada; Kiyosei Takasu
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, Oct. 2016, [Reviewed] - Desymmetrization of acid anhydride with asymmetric esterification catalyzed by chiral phosphoric acid
Ken-ichi Yamada; Akinori Oonishi; Yusuke Kuroda; Shingo Harada; Hiroki Kiyama; Yousuke Yamaoka; Kiyosei Takasu
TETRAHEDRON LETTERS, Sep. 2016, [Reviewed] - Striking Difference between Succinimidomethyl and Phthalimidomethyl Radicals in Conjugate Addition to Alkylidenemalonate Initiated by Dimethylzinc
Ken-ichi Yamada; Yusuke Matsumoto; Shintaro Fujii; Takehito Konishi; Yousuke Yamaoka; Kiyosei Takasu
JOURNAL OF ORGANIC CHEMISTRY, May 2016, [Reviewed] - Oxa- and Azacycle Formation via Migrative Cyclization of Sulfonylalkynol and Sulfonylalkynamide with N-Heterocyclic Carbene
Yinli Wang; Raphael Oriez; Satoru Kuwano; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
JOURNAL OF ORGANIC CHEMISTRY, Mar. 2016, [Reviewed] - Asymmetric Total Synthesis of Tylophorine through a Formal [2+2] Cycloaddition Followed by Migrative Ring Opening of a Cyclobutane
Yousuke Yamaoka; Marie Taniguchi; Ken-ichi Yamada; Kiyosei Takasu
SYNTHESIS-STUTTGART, Sep. 2015, [Reviewed] - An Arylative Ring Expansion Cascade of Fused Cyclobutenes via Short-Lived Intermediates with Planar Chirality
Norihito Arichi; Ken-ichi Yamada; Yousuke Yamaoka; Kiyosei Takasu
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, Aug. 2015, [Reviewed] - Organocatalytic Activation of the Leaving Group in the Intramolecular Asymmetric S(N)2 ' Reaction
Yusuke Kuroda; Shingo Harada; Akinori Oonishi; Yousuke Yamaoka; Ken-ichi Yamada; Kiyosei Takasu
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, Jul. 2015, [Reviewed] - Contiguous radical pivaloyloxymethylation-directed C(sp(3))-H iodination of N-tosyl cycloalkanecarbaldimine
Shintaro Fujii; Mayu Nakano; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada; Kiyoshi Tomioka
TETRAHEDRON LETTERS, Jun. 2015, [Reviewed] - Hydrostannylation-Cross-Coupling Strategy for the Stereoselective Synthesis of Alkylidenemalonates and Related alpha,beta-Unsaturated Esters
Shinichi Fujiwara; Romain Cadou; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, Feb. 2015, [Reviewed] - N-Heterocyclic Carbene-Catalyzed Benzoin Strategy for Divergent Synthesis of Cyclitol Derivatives from Alditols
Bubwoong Kang; Toshiaki Sutou; Yinli Wang; Satoru Kuwano; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
ADVANCED SYNTHESIS & CATALYSIS, Jan. 2015, [Reviewed] - Synthesis of steroidal derivatives bearing a small ring using a catalytic [2+2] cycloaddition and a ring-contraction rearrangement
Norihito Arichi; Kenji Hata; Yoshiji Takemoto; Ken-ichi Yamada; Yousuke Yamaoka; Kiyosei Takasu
TETRAHEDRON, Jan. 2015, [Reviewed] - Development of a Bronsted Acid-Promoted Arene-Ynamide Cyclization toward the Total Syntheses of Marinoquinolines A and C and Aplidiopsamine A
Yousuke Yamaoka; Takahiro Yoshida; Makiko Shinozaki; Ken-ichi Yamada; Kiyosei Takasu
JOURNAL OF ORGANIC CHEMISTRY, Jan. 2015, [Reviewed] - Radical Aminomethylation of Imines
Shintaro Fujii; Takehito Konishi; Yusuke Matsumoto; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
JOURNAL OF ORGANIC CHEMISTRY, Sep. 2014, [Reviewed] - Equilibration of the [2+2] Cycloaddition of Silyl Enol Ethers Catalyzed by Ethylaluminium Dichloride: Diastereoselectivity Switch in the Synthesis of Fused Cyclobutanes
Kenji Hata; Norihito Arichi; Yousuke Yamaoka; Ken-ichi Yamada; Yoshiji Takemoto; Kiyosei Takasu
ASIAN JOURNAL OF ORGANIC CHEMISTRY, Jun. 2014, [Reviewed] - Synthesis of Functionalized Polycyclic Aromatic Compounds via a Formal [2+2]-Cycloaddition
Yuuki Nagamoto; Yousuke Yamaoka; Shun Fujimura; Yoshiji Takemoto; Kiyosei Takasu
ORGANIC LETTERS, Feb. 2014, [Reviewed] - Catalytic [2+2] Cycloaddition of Silyl Enol Ethers
Yamaoka Y; Takasu K
Methods and Applications of Cycloaddition Reactions in Organic Syntheses, 2014, [Reviewed] - Kinetic Resolution of Secondary Alcohols Catalyzed by Chiral Phosphoric Acids
Shingo Harada; Satoru Kuwano; Yousuke Yamaoka; Ken-ichi Yamada; Kiyosei Takasu
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, Sep. 2013, [Reviewed] - Enhanced Rate and Selectivity by Carboxylate Salt as a Basic Cocatalyst in Chiral N-Heterocyclic Carbene-Catalyzed Asymmetric Acylation of Secondary Alcohols
Satoru Kuwano; Shingo Harada; Bubwoong Kang; Raphael Oriez; Yousuke Yamaoka; Kiyosei Takasu; Ken-ichi Yamada
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, Aug. 2013, [Reviewed] - Synthesis of 2,3,4,5-tetra-substituted pyrroles via a base-promoted double Michael reaction of oxime-enoates with nitroolefins
Yusuke Kuroda; Kazuto Imaizumi; Ken-Ichi Yamada; Yosuke Yamaoka; Kiyosei Takasu
Tetrahedron Letters, Jul. 2013, [Reviewed] - Rapid Total Syntheses Utilizing "Supersilyl" Chemistry
Brian J. Albert; Yousuke Yamaoka; Hisashi Yamamoto
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2011, [Reviewed] - Super Silyl Stereo-Directing Groups for Complete 1,5-Syn and -Anti Stereoselectivities in the Aldol Reactions of beta-Siloxy Methyl Ketones with Aldehydes
Yousuke Yamaoka; Hisashi Yamamoto
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, Apr. 2010, [Reviewed] - Chiral-thiourea-catalyzed direct Mannich reaction
Yousuke Yamaoka; Hideto Miyabe; Yoshizurm Yasui; Yoshiji Takemoto
SYNTHESIS-STUTTGART, Aug. 2007, [Reviewed] - Catalytic enantioselective petasis-type reaction of quinolines catalyzed by a newly designed thiourea catalyst
Yousuke Yamaoka; Hideto Miyabe; Yoshiji Takemoto
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, May 2007, [Reviewed] - Reactive ketimino radical acceptors: Intermolecular alkyl radical addition to imines with a phenolic hydroxyl group
H Miyabe; Y Yamaoka; Y Takemoto
JOURNAL OF ORGANIC CHEMISTRY, Mar. 2006, [Reviewed] - Triethylborane-induced intermolecular radical addition to ketimines
H Miyabe; Y Yamaoka; Y Takemoto
JOURNAL OF ORGANIC CHEMISTRY, Apr. 2005, [Reviewed] - Aqueous medium radical addition to ketimines with a phenolic hydroxyl group
H Miyabe; Y Yamaoka; Y Takemoto
SYNLETT, Nov. 2004, [Reviewed] - Palladium-indium iodide-mediated allylation and propargylation of glyoxylic oxime ether and hydrazone: The role of water in directing the diastereoselective allylation
H Miyabe; Y Yamaoka; T Naito; Y Takemoto
JOURNAL OF ORGANIC CHEMISTRY, Feb. 2004, [Reviewed] - Regioselectivity in palladium-indium iodide-mediated allylation reaction of glyoxylic oxime ether and N-sulfonylimine
H Miyabe; Y Yamaoka; T Naito; Y Takemoto
JOURNAL OF ORGANIC CHEMISTRY, Aug. 2003, [Reviewed]
MISC
- Synthesis of π-extended benzofurans via acid induced retro [2+2] cycloaddition
高須清誠; 長尾高明; 黒川宗希; 小川直希; 黒田悠介; 山岡庸介; 瀧川紘
日本薬学会年会要旨集(Web), 2023 - Synthesis and studies of isolable medium-sized (1Z,3E)-cycloalkadiene platinum complexes
紀之内颯; 伊藤智裕; 黒田悠介; 山岡庸介; 瀧川紘; 高須清誠
日本薬学会年会要旨集(Web), 2023 - ABCトランスポーターとの共結晶形成を指向したローダミン誘導体の合成と評価
三和空知; 瀧川紘; 竹内莉奈; 小田島圭; 水沼諒; 山岡庸介; 潘東青; 加藤博章; 高須清誠
次世代を担う有機化学シンポジウム講演要旨集, 2022 - Benzyne platform for intramolecular ene reaction, part 2: Application to expeditious synthesis of highly functionalized allenamides
田渡司; 加藤律希; 山岡庸介; 高須清誠; 瀧川紘
日本薬学会年会要旨集(Web), 2022 - Benzyne platform for intramolecular ene reaction, part 1: Application to stereoselective arylation of allyl alcohols
瀧川紘; 加藤律希; 田渡司; 山岡庸介; 高須清誠
日本薬学会年会要旨集(Web), 2022 - Synthesis and optical properties of helicene-xanthene hybrid dyes
三和空知; 水谷大地; 山岡庸介; 高須清誠; 瀧川紘
日本薬学会年会要旨集(Web), 2022 - Photoinduced domino reaction of ynamide leading to N-heterocycles
山岡庸介; 梶原大悟; 瀧川紘; 高須清誠
日本薬学会年会要旨集(Web), 2022 - Synthesis and Chromic properties of Hydroxyfluoranthenes
黒川宗希; 小川直希; 山岡庸介; 瀧川紘; 高須清誠
日本薬学会年会要旨集(Web), 2022 - Total Synthesis of Cryptopleurine Derivatives and their Bioactivity Evaluation
山岡庸介; 立石海斗; 山川拓朗; 服部明; 瀧川紘; 掛谷秀昭; 高須清誠
日本薬学会年会要旨集(Web), 2021 - Asymmetric Induction in the Intramolecular Migrative Cyclization of Propargylsulfones
山崎航太; 山内映穂; 宮川泰典; 猪熊翼; 山岡庸介; 高須清誠; 山田健一
日本薬学会年会要旨集(Web), 2021 - Expeditious synthesis of dibromo-ortho-quinonemonoacetals via bromination/dearomaization sequence
瀧川紘; 林隼矢; 大山侃志; 山岡庸介; 高須清誠
日本薬学会年会要旨集(Web), 2021 - Oxidative β-cleavage of a cyclobutane ring of polycyclic cyclobutanols
高須清誠; 紀之内颯; 山岡庸介; 瀧川紘
日本薬学会年会要旨集(Web), 2021 - 2-(Chlorodiisopropylsilyl)-6-(trimethylsilyl)phenyl Triflate: A Novel Platform for Intramolecular Benzyne Reactions
瀧川紘; 田渡司; 山岡庸介; 高須清誠
日本薬学会年会要旨集(Web), 2021 - Structure-ATPase activity relationship of rhodamine derivatives as transport substrates for P-glycoprotein CmABCB1
瀧川紘; 三和空知; 山岡庸介; 山口知宏; 中津亨; 加藤博章; 高須清誠
日本薬学会年会要旨集(Web), 2020 - カリウム塩基を用いる分子内エノラート-オレフィンメタセシス
高須清誠; 杉本和馬; 藤村駿; 紀之内颯; 宮川泰典; 山田健一; 瀧川紘; 山岡庸介
次世代を担う有機化学シンポジウム講演要旨集, 2020 - Intramolecular [3+2] cycloaddition of benzyne with heteroatom-substituted alkynes
瀧川紘; 田渡司; 山岡庸介; 高須清誠
日本薬学会年会要旨集(CD-ROM), 2020 - Asymmetric oxacycle-formation via migrative cyclization of sulfonylalkynol using chiral counter cation catalyst
山崎航太; 山内映穂; 宮川泰典; 猪熊翼; 山岡庸介; 高須清誠; 山田健一
日本薬学会年会要旨集(CD-ROM), 2020 - Total Synthesis of Cryptopleurine Derivatives and their Activity Evaluation
山岡庸介; 山川拓朗; 服部明; 瀧川紘; 高須清誠
日本薬学会年会要旨集(CD-ROM), 2020 - Total synthesis of an antiviral neolignan (+)-helisorin
瀧川紘; 大山侃志; 山岡庸介; 高須清誠
日本薬学会年会要旨集(CD-ROM), 2020 - An efficient synthesis of spiroindolines using ynamides
山岡庸介; 山崎大資; 梶原大悟; 瀧川紘; 高須清誠
日本薬学会年会要旨集(CD-ROM), 2020 - Synthesis and structure-ATPase activity relationship of rhodamine derivatives against P-glycoprotein CmABCB1
瀧川紘; 三和空知; 竹内莉奈; 山岡庸介; PAN Dongqing; 中津亨; 加藤博章; 高須清誠
複素環化学討論会講演要旨集, 2020 - 不斉補助基を活用したオルトキノンモノアセタールに対する立体選択的1,2-付加反応の開発
瀧川紘; 野々上喜一; 阪田慶一郎; 大山侃志; 山岡庸介; 鈴木啓介; 高須清誠
日本薬学会年会要旨集(CD-ROM), 2019 - 抗ウイルス性化合物ヘリソリンの合成研究
大山侃志; 野々上喜一; 山岡庸介; 瀧川紘; 高須清誠
日本分析化学会有機微量分析研究懇談会・計測自動制御学会力学量計測部会合同シンポジウム講演要旨集, 2019 - エンイナミドの連続環化反応による多環性キノリンの合成開発
山崎大資; 瀧川紘; 山岡庸介; 高須清誠
日本分析化学会有機微量分析研究懇談会・計測自動制御学会力学量計測部会合同シンポジウム講演要旨集, 2019 - 新規光学活性オルトキノンモノアセタールの開発と天然物合成への応用
瀧川紘; 野々上喜一; 大川侃志; 阪田慶一郎; 山岡庸介; 鈴木啓介; 高須清誠
次世代を担う有機化学シンポジウム講演要旨集, 2019 - エン‐イナミドを用いた含窒素複素環の合成法の開発と応用
山岡庸介; 山崎大資; 篠崎麻紀子; 武内奈央; 山田健一; 瀧川紘; 高須清誠
反応と合成の進歩シンポジウム講演要旨集, 15 Oct. 2018 - キラルNHC触媒を用いるα‐ヒドロキシカルボン酸誘導体の速度論的光学分割
山田健一; WANG Yinli; 猪熊翼; 山岡庸介; 高須清誠
日本プロセス化学会サマーシンポジウム講演要旨集, 02 Jul. 2018 - キラルNHC触媒を用いるキラル第二級アルコール類の速度論的光学分割とアキラルカルボン酸の添加効果
山田健一; WANG Yinli; 鍬野哲; 猪熊翼; 山岡庸介; 高須清誠
シンポジウム「モレキュラー・キラリティー」講演要旨集, 11 May 2018 - 電子環状反応を利用したtrans‐シクロアルケンの新規合成法とその応用
伊藤智裕; 堤正貴; 瀧川紘; 山田健一; 山岡庸介; 高須清誠
シンポジウム「モレキュラー・キラリティー」講演要旨集, 11 May 2018 - Synthesis of Protoilludanes Regulating Plant Growth
下田和摩; 山岡庸介; 瀧川紘; 山田健一; 高須清誠
天然有機化合物討論会講演要旨集(Web), 2018 - 基質と共触媒との水素結合複合体形成を基盤とするα‐ヒドロキシチオアミドの速度論的光学分割法の開発
王胤力; 王胤力; 山内映穂; 猪熊翼; 山岡庸介; 高須清誠; 山田健一
日本薬学会年会要旨集(CD-ROM), 2018 - キラルNHC触媒を用いる不斉アシル化によるα‐ヒドロキシカルボン酸誘導体の速度論的光学分割
王胤力; 王胤力; 猪熊翼; 山岡庸介; 高須清誠; 山田健一
反応と合成の進歩シンポジウム講演要旨集, 16 Oct. 2017 - Efficient Synthesis of Polyaromatic Hydrocarbon via a Formal [2+2] Cycloaddition
Yousuke Yamaoka
YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, Nov. 2016 - スルホニルアルキノールとスルホニルアルキンアミドのスルホニル基転位を伴う環化反応
WANG Yinli; WANG Yinli; 宮川泰典; ORIEZ Raphaeel; 山岡庸介; 高須清誠; 山田健一
複素環化学討論会講演要旨集, 09 Sep. 2016 - キラルリン酸による触媒的求核置換反応を用いるアミノアルコールの速度論的光学分割
黒田悠介; 原田慎吾; 木山大樹; 大西亨典; 山岡庸介; 高須清誠; 山田健一
日本薬学会年会要旨集(CD-ROM), 2016 - 求電子種の活性化に基づく触媒的不斉置換反応の開発
KURODA YUSUKE; HARADA SHINGO; ONISHI YUKINORI; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
次世代を担う有機化学シンポジウム講演要旨集, 22 May 2015 - Enantioselective Intermolecular [2+2] Photocycloaddition Reaction
Yousuke Yamaoka
JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN, Feb. 2015 - Synthetic Study of Cyclitols Using Benzoin-type Cyclization of Dialdoses
Kang Bubwoong; Yamaoka Yousuke; Takasu Kiyosei; Yamada Ken-ichi
Symposium on the Chemistry of Natural Products, symposium papers, 2015 - 非対称アルキリデンマロネートの立体選択的合成法のワンポット化とその応用
YAMADA KEN'ICHI; FUJIWARA SHIN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2015 - イナミドを用いたキノリン骨格の効率的合成法の開発とAplidiopsamine Aの全合成
YAMAOKA YOSUKE; SHINOZAKI MAKIKO; YOSHIDA TAKUHIRO; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2015 - 非対称ジアルドースのベンゾイン型環化反応
KAN NORIO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
日本薬学会年会要旨集(CD-ROM), 2015 - N‐トシルイミンへのラジカル付加反応に続くC(sp3)‐Hヨウ素化反応
FUJII SHINTARO; NAKANO MAYU; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI; TOMIOKA KIYOSHI
日本薬学会年会要旨集(CD-ROM), 2015 - NHCを用いるスルホニルアルキノールのスルホニル基転位を伴う環化反応
YAMADA KEN'ICHI; O INRIKI; RAPHAEL ORIEZ; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2015 - 面性不斉短寿命中間体を経る縮環シクロブテンの環拡大反応
ARICHI NORITO; YAMADA KEN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2015 - 脱離基の活性化に基づく触媒的分子内不斉SN2’反応の開発
KURODA YUSUKE; HARADA SHINGO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
反応と合成の進歩シンポジウム講演要旨集, 22 Oct. 2014 - 縮環シクロブタノールの環縮小転位を利用したtylophorine類の合成
TANIGUCHI MARIE; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
複素環化学討論会講演要旨集, 25 Aug. 2014 - 縮環シクロブタノールを経る多環芳香族化合物の合成と反応機構
YAMAOKA YOSUKE; FUJIMURA SHUN; NAGAMOTO YUKI; YAMADA KEN'ICHI; TAKASU KIYOSEI
基礎有機化学討論会要旨集, 25 Aug. 2014 - アルキリデンマロネートおよび類縁体のE/Z選択的な合成法の開発
FUJIWARA SHIN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
日本プロセス化学会サマーシンポジウム講演要旨集, 01 Jul. 2014 - 効率的縮環シクロブタノール合成と多環芳香族炭化水素への応用
YAMAOKA YOSUKE; FUJIMURA SHUN; NAGAMOTO YUKI; KISHIDA ASUMI; YAMADA KEN'ICHI; TAKEMOTO YOSHIJI; TAKASU KIYOSEI
次世代を担う有機化学シンポジウム講演要旨集, 23 May 2014 - Total Synthesis of Antitumor Terpene Paesslerin A Using Multi-component Cascade Reaction
Mogi Yuzo; Inanaga Kazato; Ishii Takayuki; Tokuyama Hidetoshi; Ihara Masataka; Yamaoka Yousuke; Yamada Ken-ichi; Takasu Kiyosei
Symposium on the Chemistry of Natural Products, symposium papers, 2014 - 縮環シクロブタノールを鍵中間体とするtylophorine類の合成研究
TANIGUCHI MARIE; YAMADA KEN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - イナミドを用いた効率的中員環合成法の開発
YAMAOKA YOSUKE; TAKEUCHI NAO; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - 2‐アシル‐2’‐アルケニルビアリールの形式的[2+2]環化付加の反応機構に関する研究
YAMAOKA YOSUKE; FUJIMURA SHUN; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - 多成分連続反応を利用するプロトイルダン類の合成研究
MOGI YUZO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - NHCを用いるスルホニルアルキノールのスルホニル基転位を伴う環状エーテル形成反応
O INRYOKU; YAMADA KEN'ICHI; ORIEZ RAPHAEEL; O SHOGUN; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - キラルリン酸触媒によるσ対称酸無水物の非対称化
YAMAOKA YOSUKE; ONISHI YUKINORI; HARADA SHINGO; KURODA YUSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - 脱離基の活性化に基づく触媒的分子内不斉SN2’反応の開発
KURODA YUSUKE; HARADA SHINGO; YAMADA KEN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2014 - D環側鎖の配座制御を志向した小員環を有するステロイド類の合成
ARICHI NORIHITO; HATA KENJI; YAMADA KEN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
有機合成シンポジウム講演要旨集, 28 Oct. 2013 - ジアルドースの立体選択的ベンゾイン環化による光学活性シクリトール類の合成
KYO NORIO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
反応と合成の進歩シンポジウム講演要旨集, 15 Oct. 2013 - 反応集積化によるプロトイルダン類の合成研究
MOGI YUZO; INANAGA KAZATO; ISHII TAKAYUKI; TOKUYAMA HIDETOSHI; IHARA MASATAKA; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
香料・テルペンおよび精油化学に関する討論会講演要旨集, 05 Oct. 2013 - アミノメチルラジカルのイミンへの付加反応
FUJII SHINTARO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
複素環化学討論会講演要旨集, 01 Oct. 2013 - 触媒的アシル化によるcis‐アリールシクロヘキサノールの速度論的光学分割
HARADA SHINGO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本プロセス化学会サマーシンポジウム講演要旨集, 21 Jun. 2013 - NHC触媒を用いるジオール及びアミノアルコール類の速度論的光学分割
KUWANO TETSU; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
次世代を担う有機化学シンポジウム講演要旨集, 24 May 2013 - キラルリン酸による触媒的アシル化:アルコールの速度論的光学分割
HARADA SHINGO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
シンポジウム「モレキュラー・キラリティー」講演要旨集, 10 May 2013 - 水素結合を利用するキノン/ヒドロキノン類の構造変化に関する研究
TAKASU KIYOSEI; NISHINO WATARU; YAMAOKA YOSUKE; YAMADA KEN'ICHI
日本薬学会年会要旨集(CD-ROM), 2013 - キラルN‐アルコキシカルボニルイミンを用いる光学活性N‐メチルアミン合成法の開発
YAMADA KEN'ICHI; YATANI TAIKI; FUJII SHINTARO; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2013 - キラルブレンステッド酸触媒を用いたアシル化による第二級アルコールの速度論的光学分割
HARADA SHINGO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2013 - クロスカップリング反応を用いるE/Z選択的アルキリデンマロネート類合成法の開発
YAMADA KEN'ICHI; FUJIWARA SHIN'ICHI; YAMAOKA YOSUKE; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2013 - イナミドを用いたキノリン骨格の効率的合成法の開発と天然物合成への応用
YAMAOKA YOSUKE; YOSHIDA TAKAHIRO; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2013 - 膜タンパク質変性作用の少ない可溶化剤の開発
HAYASHIDA KOICHI; MOGI YUZO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YANO YOSHIAKI; MATSUZAKI KATSUMI
日本薬学会年会要旨集(CD-ROM), 2013 - シクロブタノール形成反応を利用する多環芳香族炭化水素の合成
TAKASU KIYOSEI; NAGAMOTO YUKI; KISHIDA ASUMI; YAMADA KEN'ICHI; YAMAOKA YOSUKE
日本薬学会年会要旨集(CD-ROM), 2013 - カルボン酸の添加によるキラルNHC触媒を用いる第2級アルコールの速度論的光学分割の反応加速と選択性向上
KUWANO SATORU; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
日本薬学会年会要旨集(CD-ROM), 2013 - D環側鎖の配座制御を志向した小員環を有するエストロン誘導体の合成
ARICHI NORIHITO; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集(CD-ROM), 2013 - 新規連続的8π-6π電子環状反応を利用した多環性縮環シクロブタノールの構築と多環芳香族化合物合成への応用
永本祐樹; 岸田明日美; 山岡庸介; 竹本佳司; 高須清誠
第102回有機合成シンポジウム, Nov. 2012, [Reviewed] - 連続的8π‐6π電子環状反応を利用する多環性シクロブタノールの立体制御合成
YAMAOKA YOSUKE; KISHIDA ASUMI; NAGAMOTO YUKI; YAMADA KEN'ICHI; TAKEMOTO YOSHIJI; TAKASU KIYOSEI
反応と合成の進歩シンポジウム講演要旨集, 15 Oct. 2012 - キラルNHC触媒を用いる第2級アルコールの速度論的光学分割の開発
KUWANO SATORU; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
反応と合成の進歩シンポジウム講演要旨集, 15 Oct. 2012 - イナミドを用いた多環性キノリン合成法の開発
YAMAOKA YOSUKE; YOSHIDA TAKAHIRO; YAMADA KEN'ICHI; TAKASU KIYOSEI
複素環化学討論会講演要旨集, 30 Sep. 2012 - 対称ジアルデヒドの分子内不斉ベンゾイン縮合と光学活性シクリトール類合成への応用
KYO NORIO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
有機合成化学セミナー講演予稿集, 05 Sep. 2012 - アルキリデンマロネートのオキシメチル化反応の制御
YAMADA KEN'ICHI; KONISHI TAKETO; NAKANO MAYU; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMAMOTO YASUTOMO; TOMIOKA KIYOSHI
有機合成化学セミナー講演予稿集, 05 Sep. 2012 - 連続的8π‐6π電子環状反応による多環性シクロブタノールの合成
KISHIDA ASUMI; NAGAMOTO YUKI; TAKEMOTO YOSHIJI; YAMAOKA YOSUKE; YAMADA KEN'ICHI; TAKASU KIYOSEI
日本薬学会年会要旨集, 05 Mar. 2012 - α‐アミノアルキルラジカルのイミンへの付加反応の開発
FUJII SHINTARO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
日本薬学会年会要旨集, 05 Mar. 2012 - C2対称ジアルデヒドのベンゾイン縮合による光学活性シクリトール類の合成
KYO NORIO; YAMAOKA YOSUKE; TAKASU KIYOSEI; YAMADA KEN'ICHI
日本薬学会年会要旨集, 05 Mar. 2012 - Aldol Methodologies Utilizing Super Silyl Groups for Polyketide Synthesis
Hisashi Yamamoto; Brian J. Albert; Yousuke Yamaoka
SYNTHESIS-STUTTGART, Jul. 2010
Books and other publications
Lectures, oral presentations, etc.
- エン-イナミドを用いた含窒素複素環の合成法の開発と応用
山岡 庸介
第44回反応と合成の進歩シンポジウム, Nov. 2018 - ブレンステッド酸によるイナミドの分子内スピロ環化反応の開発
山岡 庸介
第68回日本薬学会近畿支部総会・大会, Oct. 2018 - イナミドを用いた新規スピロインドリン合成法の開発
山岡 庸介
日本薬学会第138年会, Mar. 2018 - ケテンシリルアセタールの触媒的(2+2)環化付加によるシクロブテンの合成
山岡 庸介
日本プロセス化学会2017サマーシンポジウム, Aug. 2017 - イナミドを用いた含窒素複素環合成
山岡 庸介
イナミドを用いた含窒素複素環合成, Jun. 2017, [Invited] - エン‐イナミドを用いた含窒素複素環の簡便合成法の開発と応用
山岡 庸介
第42回反応と合成の進歩シンポジウム, Nov. 2016 - 形式的[2+2]環化反応を用いた多環芳香族炭化水素の合成とその応用
山岡 庸介
第66回日本薬学会近畿支部総会, Oct. 2016, [Invited] - ケテンシリルアセタールとプロピオール酸エステルの触媒的[2+2]環化付加反応の開発
山岡 庸介
第46回複素環化学討論会, Sep. 2016 - イナミドを用いたキノリン骨格の効率的合成法の開発とAplidiopsamine Aの全合成
山岡 庸介
第135回日本薬学会年会, Mar. 2015 - イナミドを用いた中員環の効率的合成法の開発
山岡 庸介
第64回日本薬学会近畿支部総会, Oct. 2014 - 効率的縮環シクロブタノール合成と多環芳香族炭化水素への応用
山岡 庸介
第12回次世代を担う有機化学シンポジウム, May 2014 - イナミドを用いた効率的中員環合成法の開発
山岡 庸介
Mar. 2014 - Marinoquinoline類およびAplidiopsamine Aの全合成
山岡 庸介
第63回日本薬学会近畿支部総会, Oct. 2013 - Base-Induced Stereoselective Formation of Benzo-fused Cyclobutanols from Biarylketones
山岡 庸介
ISCC-10, Sep. 2013, [Invited] - イナミドを用いたキノリン骨格の効率的合成法の開発と天然物合成への応用
山岡 庸介
第133回日本薬学会年会, Feb. 2013
Research Themes
- Efficient Synthesis of Cyclobutanes by Multicomponent Reaction Using Ynolates and Its Application for Drug Discovery
Grant-in-Aid for Scientific Research (C)
Hyogo Medical University
Apr. 2024 - Mar. 2027 - Design, Synthesis and Evaluation of Biologically Active Molecules Based on Ring Strain
Grant-in-Aid for Scientific Research (B)
Kyoto University
Apr. 2019 - Mar. 2022 - Divergent Synthesis of Nitrogen-Containing Heterocycles by Sequential Reactions and Its Application to Drug Discovery
Grant-in-Aid for Scientific Research (C)
Kyoto University
Apr. 2018 - Mar. 2021 - Stereocontrolled synthesis of poly-substituted medium-sized cyclic compounds by electrocyclic ring opening reaction and the synthesis of biologically active molecules
Grant-in-Aid for Scientific Research (B)
Kyoto University
Apr. 2016 - Mar. 2019 - Efficient synthesis of nitrogen-containing compounds with yanamides
Grant-in-Aid for Young Scientists (B)
Kyoto University
Apr. 2016 - Mar. 2018 - Discovery of new reactions and utilities of 4-membered carbocyles based on their unique ring strains.
Grant-in-Aid for Scientific Research (B)
Kyoto University
Apr. 2013 - Mar. 2016 - Development of a Bronsted Acid-Promoted Ene-Ynamide Cyclization
Grant-in-Aid for Young Scientists (B)
Kyoto University
Apr. 2013 - Mar. 2015